BISOPROLOL

Bisoprolol is a selective beta-1 adrenergic blocker used to manage hypertension and heart failure. It works by reducing heart rate and blood pressure, thereby decreasing the workload on the heart. Bisoprolol is typically administered orally in tablet form. It can also be used to treat chronic stable angina and certain types of arrhythmias. Common side effects include fatigue, dizziness, and cold extremities. It should be used cautiously in patients with respiratory conditions or diabetes.

Bisoprolol is a medication that belongs to the class of beta-blockers. Here is a detailed description:

Chemical Name: 1-[4-[[2-(1-Methylethoxy)ethoxy]methyl]phenoxy]-3-(1-methylethylamino)propan-2-ol

Molecular Formula: C18H31NO4

Mechanism of Action:

  • Bisoprolol works by blocking beta-1 adrenergic receptors, reducing heart rate, and decreasing blood pressure.

Indications:

  • Hypertension (high blood pressure)
  • Heart failure
  • Angina pectoris (chest pain)

Pharmacokinetics:

  • Absorption: Well absorbed after oral administration
  • Distribution: Widely distributed throughout the body
  • Metabolism: Metabolized in the liver
  • Excretion: Excreted in the urine

Side Effects:

  • Fatigue
  • Dizziness
  • Headache
  • Nausea and vomiting
  • Bradycardia (slow heart rate)

Contraindications:

  • Hypersensitivity to Bisoprolol
  • Severe bradycardia
  • Heart block
  • Cardiogenic shock
  • Severe asthma
  • Pregnancy (caution)

Dosage: avoid self medication

  • Oral: 2.5-20 mg, once daily

Forms:

  • Tablets

Please note that this information is not a substitute for medical advice. If you have any questions or concerns about Bisoprolol or any other medication, please consult a healthcare professional.