Disease Related

METOPROLOL

Metoprolol is a selective beta-1 adrenergic blocker used to treat various cardiovascular conditions, including hypertension, angina, and heart failure. It works by reducing heart rate and blood pressure, which decreases the heart’s workload. Metoprolol is typically administered orally in tablet form, but it can also be given intravenously in hospital settings. Common side effects include fatigue, dizziness, and cold hands or feet. It should be used with caution in individuals with respiratory conditions, diabetes, or certain heart conditions.

Metoprolol is a medication that belongs to the class of beta-blockers. Here is a detailed description:

Chemical Name: 1-[4-(2-methoxyethyl)phenoxy]-3-[(1-methylethyl)amino]propan-2-ol

Molecular Formula: C15H25NO3

Mechanism of Action:

  • Metoprolol works by blocking beta-1 adrenergic receptors, reducing heart rate, and decreasing blood pressure.

Indications:

  • Hypertension (high blood pressure)
  • Angina pectoris (chest pain)
  • Heart failure
  • Cardiac arrhythmias (abnormal heart rhythms)
  • Myocardial infarction (heart attack)

Pharmacokinetics:

  • Absorption: Well absorbed after oral administration
  • Distribution: Widely distributed throughout the body
  • Metabolism: Metabolized in the liver
  • Excretion: Excreted in the urine

Side Effects:

  • Fatigue
  • Dizziness
  • Headache
  • Nausea and vomiting
  • Bradycardia (slow heart rate)

Contraindications:

  • Hypersensitivity to Metoprolol
  • Severe bradycardia
  • Heart block
  • Cardiogenic shock
  • Severe asthma
  • Pregnancy (caution)

Dosage: avoid self medication

  • Oral: 25-400 mg, every 12 hours

Forms:

  • Tablets
  • Extended-release tablets
  • Injection

Please note that this information is not a substitute for medical advice. If you have any questions or concerns about Metoprolol or any other medication, please consult a healthcare professional.