Chemical Name: 5-[1-hydroxy-2-[(1-methyl-3-phenylpropyl)amino]ethyl]salicylamide
Molecular Formula: C19H24N2O3
Mechanism of Action:
- Labetalol works by blocking both alpha- and beta-adrenergic receptors, reducing blood pressure and heart rate.
Indications:
- Hypertension (high blood pressure)
- Severe hypertension (emergency situations)
Pharmacokinetics:
- Absorption: Well absorbed after oral administration
- Distribution: Widely distributed throughout the body
- Metabolism: Metabolized in the liver
- Excretion: Excreted in the urine
Side Effects:
- Fatigue
- Dizziness
- Headache
- Nausea and vomiting
- Hypotension (low blood pressure)
Contraindications:
- Hypersensitivity to Labetalol
- Severe bradycardia
- Heart block
- Cardiogenic shock
- Severe asthma
- Pregnancy (caution)
Dosage: avoid self medication
- Oral: 100-800 mg, every 12 hours
- Intravenous: 20-80 mg, every 10-30 minutes
Forms:
- Tablets
- Injection
Please note that this information is not a substitute for medical advice. If you have any questions or concerns about Labetalol or any other medication, please consult a healthcare professional.